庫存單位: PKSH033982_10μg-ES

重組人 BRD4 (N-10His-Flag),10 μg

溴結構域蛋白 4 (BRD4) 是 BET 類染色質讀取蛋白的成員,可結合乙醯化組蛋白並在轉錄調控和表觀遺傳記憶傳遞中發揮關鍵作用。在整個細胞週期中與乙醯化染色質保持相關,並透過保存乙醯化染色質狀態和維持高級染色質結構為有絲分裂後 G1 基因轉錄提供表觀遺傳記憶。 BRD 溴結構域作為組蛋白上乙醯化賴氨酸殘基的識別基序,而 NET 結構域可能透過促進 RNA 聚合酶 II 的 C 端結構域 (CTD) 的磷酸化發揮作用。一些 BRD4 的特定抑制劑透過結合 Asn-140 和 Asn-433 來阻止其與乙醯化組蛋白的結合,是治療白血病的有希望的治療分子。 BRD4 是許多疾病的潛在治療標靶,包括乳癌、AML、多發性骨髓瘤、結腸癌等。

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Product Specification

Basic Information

Brands:Elabscience

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Place of Origin:中國

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Reconstitution:不適用

Shipping:本產品以液體形式提供。它是在冷凍溫度下用藍冰/凝膠包運輸的。收到後,立即存放在<-20°C的環境中。

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Calculated Molecular Weight:49.0 kDa

Observed Molecular Weight:55-60kDa

Purity: 以還原 SDS-PAGE 測定,結果為 > 90%。

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Storage:儲存溫度<-20°C,可穩定保存6個月。請盡量減少凍融循環。

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Calculated Molecular Weight:49.0 kDa

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Endotoxin: 經 LAL 方法測定,每 μg 蛋白質含量 < 1.0 EU。

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Research Areas:癌症;表觀遺傳學和核子訊號

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Bio-activity:未驗證活動

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Formulation:以 0.2 μm 過濾溶液的形式提供,其中含有 50mM HEPES、200mM NaCl、1mM DTT、10% 甘油,pH 7.5。

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